| Sr. No. |
Intermediate |
CAS No. |
EINECS No. |
Structure |
End use |
| Pharma Intermediates |
| 1 |
CMIC Chloride:
3-(2-Chlorophenyl)-5-methyl isoxazole-4-carbonyl chloride |
25629-50-9 |
247-137-4 |
 |
Cloxacillin |
| 2 |
DCMIC Chloride:
3-(2,6 Dichlorophenyl)-5-methyl isoxazole-4-carbonyl chloride |
4462-55-9 |
224-723-8 |
 |
Dicloxacillin |
| 3 |
FCMIC Chloride:
3-(2-Chloro-6-fluorophenyl)-5-methyl isoxazole-4-carbonyl chloride |
69399-79-7 |
273-987-0 |
 |
Flucloxacillin |
| 4 |
PMIC Chloride:
3-Phenyl-5-methyl isoxazole-4-carbonyl chloride |
16883-16-2 |
240-915-4 |
 |
Oxacillin |
| 5 |
EDPCC:
4-Ethyl-2,3-dioxopiperazine
carbonyl chloride |
59703-00-3 |
261-867-0 |
 |
Piperacillin |
| 6 |
EPCP:
(R)-[[(4-Ethyl-2,3-dioxopiperazin-1-yl)carbonyl]amino]phenylacetic acid |
63422-71-9 |
264-133-8 |
 |
Piperacillin |
7
New |
AOSA#
(3R,4R)-4-Acetoxy-3-[(R)-1-(tert-butyl-dimethylsilyloxy)ethyl]azetidin-2-one |
76855-69-1 |
408-050-9
(ELINCS) |
 |
Carbapenem |
| 8 |
Azacyclonol base:
α,α-Diphenyl-4-piperidinomethanol hydrochloride |
115-46-8 |
204-092-5 |
 |
Fexofenadine |
9
New |
Isonipecotic acid:
4-Piperidinecarboxylic acid |
498-94-2 |
207-872-3 |
 |
Fexofenadine, Risperidone |
| 10 |
GMC - XL2:
2-Deoxy-2,2-diflouro-D-erythro-pentafuranose-1-ulose-3,5-dibenzoate |
122111-01-7 |
- |
 |
Gemcitabine HCl |
| 11 |
LM3:
[1R-[1-α(2S*,5R*),2ß,5ß]]-5-(4-Amino-2-oxo-1(2H)-pyrimidinyl)-1,3-oxathiolane-2-carboxylic acid- 5-methyl-2-(1-methylethyl)cyclohexyl ester |
147126-73-6 |
- |
 |
Lamivudine |
| 12 |
1-(4-Azido-5-trityloximethyl- tetrahydrofuran-2-yl)-5-methyl-1H-pyrimidine-2,4-dione |
29706-84-1 |
- |
 |
Zidovudine |
13
New |
4-Methyl-10-trityloxymethyl-8,11-dioxa-2,6-diaza-tricyclo[7.2.1.0*2,7*] dodec-6-en-5-one |
25442-42-6 |
- |
 |
Zidovudine |
| 14 |
DKT3#:
4-Fluoro-α-(2-methyl-1-oxopropyl)-γ-oxo-N,ß-diphenyl benzene butanamide |
125971-96-2 |
- |
 |
Atorvastatin |
| 15 |
ATS-5#:
(R)-4-Cyano-3-hydroxybutyric acid ethyl ester |
141942-85-0 |
- |
 |
Atorvastatin |
| 16 |
ATS-8#:
(4R,cis)-1,1-Dimethylethyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxane-4-acetate |
125971-94-0 |
425-780-3 |
 |
Atorvastatin |
17
New |
ATS-9#:
(4R,cis)-1,1-Dimethylethyl-6-aminoethyl-2,2-dimethyl-1,3-dioxane-4-acetate |
125995-13-3 |
- |
 |
Atorvastatin |
| 18 |
ATV-1#:
tert-Butyl (4R,6R)-2-[[[6-(2-4-fluorophenyl)-5-isopropyl-3-phenyl-4-(phenylcarbamoyl)-pyrrol-1-yl]ethyl]-2,2-dimethyl-1,3-dioxan-4-yl]acetate |
125971-95-1 |
- |
 |
Atorvastatin |
19
New |
(S)-2-(2-Amino-5-chlorophenyl)-4-cyclopropyl-1,1,1-trifluoro-3-butyn-2-ol |
209414-27-7 |
- |
 |
Efavirenz |
| 20 |
Ethyl 4-chloro acetoacetate |
638-07-3 |
211-317-0 |
 |
Amlodipine |
21
New |
Ethyl 4-(2-(1,3-dioxoisoindolin-2-yl)ethoxy)-3-oxobutanoate |
88150-75-8 |
- |
 |
Amlodipine |
| 22 |
Phthaloyl amlodipine:
3-Ethyl-5-methyl-4-(2-chlorophenyl)-2-(2-phthalimidoethoxy)-methyl-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate |
88150-62-3 |
413-410-3
(ELINCS) |
 |
Amlodipine |
| 23 |
4,5,6,7-Tetrahydrothieno[3,2-c] pyridine hydrochloride |
28783-41-7 |
249-220-0 |
 |
Clopidogrel, Ticlopidine |
24
New |
Coupled amine HCl:
S-(+)-Methyl-2(2-thienylethylamino)-2-(2-chlorophenyl) acetate hydrochloride |
141109-19-5 |
- |
 |
Clopidogrel |
25
New |
Clopidogrel base:
S-(2-Chloro-phenyl)-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-acetic acid methyl ester |
113665-84-2 |
- |
 |
Clopidogrel |
| 26 |
S (-)-3-(Dimethylamino)-1-(thiophen-2-yl)propane-1-ol# |
132335-44-5 |
- |
 |
Duloxetine |
27
New |
S(-)-3-(Methylamino)-1-(thiophen-2-yl)propane-1-ol# |
116539-56-1 |
- |
 |
Duloxetine |
| 28 |
S (+) - N,N-Dimethyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl) propan-1-amine (base and oxalate)# |
132335-46-7
(Base)
132335-47-8
(Oxalate) |
- |
 |
Duloxetine |
| 29 |
DIOL#
(S)-1-[[[1-[3-[2-(7-Chloro-2-quinolinyl)ethenyl] phenyl]]-3-[2-(1-hydroxy-1-methylethyl)phenyl]propyl-1-ol]] |
142569-70-8 |
- |
 |
Montelukast |
| 30 |
AST#
(S)-2-[3-[3-[2-(7-Chloro-2-quinolinyl) ethenyl]-phenyl]-3-hydroxypropyl] benzoic acid methyl ester |
142569-69-5 |
- |
 |
Montelukast |
31
New |
Montelukast dicyclohexyl amine salt# |
- |
- |
 |
Montelukast |
| 32 |
RX5*
2-Azabicyclo[3.3.0]-octane-3-carboxylic acid benzyl ester hydrochloride |
93779-29-4 |
- |
 |
Ramipril |
| 33 |
RX7 *
(S,S,S)-2-Aza-bicyclo-[3,3,0]-octane-3-carboxylic acid benzyl ester hydrochloride |
93779-31-8 |
- |
 |
Ramipril |
| 34 |
Octahydroindol-2-carboxylic acid
(rac. 7αR/3αS/2R, 7αS/3αR/2S) |
145438-94-4 |
- |
 |
Trandolapril |
35
New |
Benzyl (2S,3αR,7αS)-octahydroindole-2-carboxylate hydrochloride |
87679-38-7 |
- |
 |
Trandolapril |
36
New |
2-Chloromethyl-3,4-dimethoxypyridine hydrochloride |
72830-09-2 |
416-440-5
(ELINCS) |
 |
Pantoprazole |
37
New |
5-(Difluromethoxy)-2-[(3-methoxy-4-chloro-2-pyridinyl)methylmercapto]-1H-benzimidazole |
368890-20-4 |
- |
 |
Pantoprazole |
38
New |
5-(Difluromethoxy)-2-[(3,4-dimethoxy-2- pyridinyl)methylmercapto]-1H-benzimidazole |
102625-64-9 |
- |
 |
Pantoprazole |
39
New |
2-[[4-(3-Methoxypropoxy)-3-methylpyridine-2-yl]methylthio]-1H-benzimidazole |
117977-21-6 |
- |
 |
Rabeprazole |
| 40 |
6-Chloro-5-(2-chloroacetyl)-2-oxyindole
|
118289-55-7 |
421-320-0
(ELINCS) |
 |
Ziprasidone |
| 41 |
6-Chloro-5-(2-chloroethyl)-2-oxyindole
|
118307-04-3 |
- |
 |
Ziprasidone |
| 42 |
3-Chloro-1,2-benzisothiazole |
7716-66-7 |
- |
 |
Ziprasidone |
43
New |
3-Piperazinyl-1,2-benzisothiazole hydrochloride |
87691-88-1 |
- |
 |
Ziprasidone |
44
New |
DIOL BASE:
4-[4-(Dimethylamino-1-(4’-fluorophenyl)1-hydroxybutyl)-3-hydroxymethyl] benzonitrile |
103146-25-4 |
- |
 |
Citalopram |
45
New |
1-(4-Chlorobenzhydryl)piperazine |
303-26-4 |
206-137-4 |
 |
Cetirizine |
46
New |
2-Thiopheneacetyl chloride
|
39098-97-0 |
254-290-0 |
 |
Cephalothine |
47
New |
2-Ethoxynaphthalene-1-carbonyl chloride |
55150-29-3 |
259-502-5 |
 |
Nafcillin |
48
New |
N-Formyl hexamethylenimine dimethyl acetal |
32895-16-2 |
32895-16-2 |
 |
Mecillinam Pivmecillinam |
49
New |
3,4-Dichloro-α methoxyphenyl acetic acid chloride |
83833-34-5 |
281-009-9 |
 |
Clometocillin |
50
New |
1,1-Cyclohexanediacetic acid mono methylester |
60142-94-1 |
- |
 |
Gabapentin |
51
New |
S(+)-2-Aminobutyramide hydrochloride |
7682-20-4 |
- |
 |
Levetiracetam |
| Specialty Chemicals / Intermediates |
| 52 |
Monomethyl acetoacetamide |
20306-75-6 |
243-723-9 |
 |
Agrochemical |
| 53 |
Aceto acetanilide |
102-01-2 |
202-996-4 |
 |
Pigment Intermediates |
54
New |
AABZ:
5-Acetoacetylaminobenzimidazol-2-one |
26576-46-5 |
247-820-7 |
 |
Pigment Intermediates |
| * Under development |
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Responsibility with respect to third party patent rights in a specific country lies exclusively with the buyer. |
| # Developed as per Codexis Inc. proprietary Biocatalysis technology |
